北海道科学大学 研究者紹介・教員紹介
English
ヤマギシ タケヒロ
Takehiro Yamagishi
山岸 丈洋
所属
北海道科学大学 薬学部 薬学科
職種
教授
著書・論文歴
著書
薬学基礎化学物理編下 京都廣川書店 (共著) 2020/03
著書
基礎有機化学問題集 (共著) 2013
論文
Synthesis of Deuterated Compounds by Flow Chemistry ChemPlusChem (共著) 2024/03/07
論文
Synthesis and structural characterization of benaene-1,3-disulfonamide-containing 11- to 13-membered heterocycles via double Mitsunobu annulation Chemistry Letters 53 (1),upad016 (共著) 2023/12/01
論文
Facile Preparation of the nootropic agent IDRA-21 and related heterocycles via a one-pot iron-mediated redox annulation Heterocycles 106 (9),1580-1588頁 (共著) 2023/08/17
論文
Divergent synthesis of benzo[
b
]phosphole oxide derivatives focusing on substituents on phosphorus atom Tetrahedron 143,133562-133567頁 (共著) 2023/07/19
論文
北海道産赤ビーツによる便通異常の改善効果についての検討 応用薬理 100 (5),95-100頁 (共著) 2021
論文
Nickel-catalyzed regio- and stereoselective hydrophosphinylation of internal ynamides with
H
-phosphinates Tetrahedron 74,7068-7073頁 (共著) 2018/10/19
論文
Copper-catalyzed Hydrophosphinylation of Terminal Ynamides with
H
-Phosphinates. Tetrahedron 73,1705-1710頁 (共著) 2017/02/09
論文
Nickel-catalyzed C-P Cross-coupling Reactions of Aryl Iodides with
H
-phosphinates. Tetrahedron 71,7614-7619頁 (共著) 2015/08/01
論文
Reductive Alkylation of Hydrazine Derivatives with α-Picoline-Borane and Its Application to the Synthesis of Useful Compounds Related to Active Pharmaceutical Ingredients. Synthesis 46,455-464頁 (共著) 2014
論文
Stereocontrolled Synthesis of Phosphinyl Dipeptide Isosteres Using an Asymmetric Center at the Phosphorus Atom. YAKUGAKU ZASSHI 134,915-924頁 (単著) 2014
論文
One-Pot Synthesis of Phenol Derivatives by the Novel Intramolecular Alder-Rickert Reaction: Effects of Aryl Substituent at the 3-Position of Cyclohexenone Derivatives on Reactivity. Chem. Pharm. Bull. 61,768-775頁 (共著) 2013
論文
Total Synthesis and Structural Revision of Incargutines A and B. Synlett 24,1998-2002頁 (共著) 2013
論文
A Safe and Scalable Procedure for Preparation of α-Picoline-Borane from Sodium Mono-acyloxyborohydrides and α-Picoline. Org. Process Res. Dev. 16,495-498頁 (共著) 2012
論文
Diastereoselective Synthesis of Pro-Phe Phosphinyl Dipeptide Isosteres. Tetrahedron: Asymmetry 23,1633-1639頁 (共著) 2012
論文
Synthesis of Phenol Derivatives from Cyclohex-2-enones Bearing an Alkyne through Lewis Acid-Catalyzed Enolization and Intramolecular Alder-Rickert Reaction. J. Org. Chem. 77,8999-9005頁 (共著) 2012
論文
A Chemo-enzymatic Synthesis of Optically Active 1,1-Diethoxyethyl(aminomethyl)phosphinates: Useful Chiral Building Blocks for Phosphinyl Dipeptide Isosteres. Tetrahedron: Asymmetry 22,1358-1363頁 (共著) 2011
論文
Diastereoselective Synthesis of the Leu-Pro Type Phosphinyl Dipeptide Isostere. J. Org. Chem. 76,5472-5476頁 (共著) 2011
論文
N
-Benzyl-Protection of Amino Acid Derivatives by Reductive Alkylation with α-Picoline-Borane. Synthesis,1673-1677頁 (共著) 2010
論文
Diastereoselective Synthesis of γ-Amino-δ-hydroxy-α,α-difluorophosphonates: A Vehicle for Structure-activity Relationship Studies on SMA-7, a Potent Sphingomyelinase Inhibitor. J. Org. Chem. 74,6350-6353頁 (共著) 2009
論文
One-pot Synthesis of Alkoxyamine Derivatives by Reductive Alkoxyamination with a 2-Picoline-borane Complex. Heterocycles 78,463-470頁 (共著) 2009
論文
Diastereoselective Synthesis of α,β'-Disubstituted Aminomethyl(2-carboxyethyl)phosphinates as Phosphinyl Dipeptide Isosteres. Org. Lett. 19,4347-4350頁 (共著) 2008
論文
Asymmetric Synthesis of Optically Active α-Substituted α-Amino-
H
-phosphinates through Resolution of 1,1-Diethoxyethyl(aminomethyl)phosphinates. Tetrahedron: Asymmetry 18,2886-2893頁 (共著) 2007
論文
Diastereoselective Addition of α-Substituted α-Amino-
H
-phosphinates to Imines Using Yb(OTf)
3
as an Efficient Lewis Acid Catalyst. Tetrahedron 63,8199-8205頁 (共著) 2007
論文
Diastereoselective Synthesis of Novel α-Amino-α'-hydroxyphosphinates by Hydrophosphinylation of α-Amino-
H
-phosphinates to Aldehydes. Synthesis,3226-3232頁 (共著) 2007
論文
Asymmetric Synthesis of Phosphonic Acid Analogues for Acylcarnitine. Tetrahedron 62,54-65頁 (共著) 2006
論文
Diastereoselective Alkylation of Iminomethylenephosphinates Possessing an Asymmetrc Center at the Phosphorus Atom. Tetrahedron 62,9210-9217頁 (共著) 2006
論文
A practical Synthesis of 8-Hydroxyacyclovir and 9-(Carboxymethoxymethyl)guanine, Metabolites of Acyclovir. Heterocycles 65,1967-1973頁 (共著) 2005
論文
Lipase-catalyzed Kinetic Resolution of α-Hydroxy-
H
-phosphinates. Tetrahedron Lett. 45,6713-6716頁 (共著) 2004
論文
Synthesis of Chiral γ-Amino-β-hydroxyphosphonate Derivatives from Unsaturated Phosphonates, Synlett,2505-2508頁 (共著) 2004
論文
Diastereoselective Synthesis of β-Substituted α-hydroxyphosphinates through Hydrophosphinylation of α-Heteroatom-substituted Aldehydes. Tetrahedron 59,767-772頁 (共著) 2003
論文
Aymmetric Synthesis of β-Amino-α-hydroxyphosphinic Acid Derivatives through Hydrophosphinylation of α-Amino Aldehydes. Tetrahedron 58,2577-2583頁 (共著) 2002
論文
Stereoselective Synthesis of β-Amino-α-hydroxy(allyl)phosphinates and an Application to the Synthesis of a Building Block for Phosphinyl Peptides. Synlett,1471-1474頁 (共著) 2002
論文
Diastereoselctive Synthesis of Chiral β-Amino-α-hydroxy-
H
-phosphinates through Hydrophosphinylation of α-Amino Aldehydes. Tetrahedron Lett 42,5033-5036頁 (共著) 2001
論文
Stereoselective Reduction of Cyclopropylalkanones Possessing a Difluoromethylenephosphonate Group at the Ring: Application to Stereoselective Synthesis of Novel Cyclopropane Nucleotide Analogues. Tetrahedron 56,7099-7108頁 (共著) 2000
論文
Conventional Synthesis of Cyclopropylalkanol Derivatives Possessing a Difluoromethylenephosphonate Group at the Ring. J. Org. Chem. 64,8413-8418頁 (共著) 1999
論文
Enantioselective Synthesis of α-Hydroxyphosphinic Acid Derivatives through Hydrophosphinylation of Aldehydes Catalyzed by Al-Li-BINOL Complex. Tetrahedron 55,12125-12136頁 (共著) 1999
論文
Asymmetric Dihydroxylation of 1-Acyloxy-2(
E
)-Alkenylphosphonates with AD-mix Reagents. Effects of 1-Acyloxy Functional Groups on the Asymmetric Dihydroxylation. Tetrahedron 54,781-790頁 (共著) 1998
論文
Enantioselective Synthesis of
threo
-α,β-Dihydroxyphosphonates by Asymmetric Dihydroxylation of 1(
E
)-Alkenylphosphonates with AD-mix Reagents. Tetrahedron 54,767-780頁 (共著) 1998
論文
Enantioselective Synthesis of α-Hydroxyphosphonates through Asymmetric Pudovik Reactions with Chiral Transition Metal Catalysts. J. Chem. Soc., Perkin Trans 1,1527-1533頁 (共著) 1997
論文
Stereocontrolled Synthesis of Hydroxymethylene Phosphonate Analogues of Phosphorylated Tyrosine and Their Conversion to Monofluoromethylene Phosphonate Analogues. Tetrahedron 52,11725-11738頁 (共著) 1996
論文
Enantioselective Synthesis of
threo
-α,β-Dihydroxyphosphonates by Asymmetric Dihydroxylation of Vinylphosphonates. An Application to the Stereocontrolled Synthesis of (4
S
,5
S
)-4-Diethylphosphono-5-hydroxymethyl-2,2-dimethyl-1,3-dioxolane. Tetrahedron: Asymmetry 6,365-368頁 (共著) 1995
論文
Highly Regioselective Silylation of α,β-Dihydroxyphosphonates: An application to Stereoselective Synthesis of α-Amino-β-hydroxyphosphonic Acid Derivatives. Synlett,847-849頁 (共著) 1995
論文
Stereoselective Synthesis of γ,δ-Unsaturated α-Hydroxyphosphonates through [2,3]-Wittig Sigmatropic Rearrangement ofα-Allyloxyphosphonates. Synlett,1035-1036頁 (共著) 1995
論文
α位にヘテロ原子団を有するホスホン酸誘導体合成の最近の進展. 有機合成化学協会誌 53,881-892頁 (共著) 1995
論文
Enantioselective Hydrophosphonylation of Aromatic Aldehydes Catalyzed by Chiral Titanium Alkoxides. Tetrahedron: Asymmetry 4,1779-1782頁 (共著) 1993
論文
Enantioselectivity for Hydrophosphonylation of Aromatic Aldehydes Catalyzed by Lanthanum Binaphthol Complex. Remarkable Electronic Effect of Aromatic Substituents. Tetrahedron: Asymmetry 4,1783-1784頁 (共著) 1993
論文
Stereodivergent Synthesis of β-Amino-α-hydroxyphosphonic Acid Derivatives by Lewis Acid Mediated Stereoselective Hydrophosphonylation of α-Amino Aldehydes. Tetrahedron: Asymmetry 4,1401-1404頁 (共著) 1993